1,2,3,4-tetrahydroquinoxaline derivatives

Intervention

1 paper1 finding

  • 1 lab in 2 countries
  • Funders: BrightFocus Foundation and 7 more
  • Cells1

Outcomes

1

NAD+

upin cells1

1 study
  1. 1,2,3,4-tetrahydroquinoxaline derivatives increase NAD+ in cells (Nanomolar potency for several compounds).

    “These findings identify tetrahydroquinoxalines as a promising class of neuronal NAD-boosting agents”

    Cellsprimary cortical neurons

    Potent Neuronal Nicotinamide Adenine Dinucleotide-Boosting Tetrahydroquinoxalines: Structure-Activity Relationships and Early Drug Metabolism and Pharmacokinetics Evaluation

    ACS medicinal chemistry letters4 Mar 2026

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