1,2,3,4-tetrahydroquinoxaline derivatives
1 paper1 finding
- 1 lab in 2 countries
- Funders: BrightFocus Foundation and 7 more
- Cells1
Outcomes
1NAD+
upin cells1
1 study
NAD+
upin cells1
1,2,3,4-tetrahydroquinoxaline derivatives increase NAD+ in cells (Nanomolar potency for several compounds).
“These findings identify tetrahydroquinoxalines as a promising class of neuronal NAD-boosting agents”
Cellsprimary cortical neurons
ACS medicinal chemistry letters4 Mar 2026
Latest
1 in 12 monthsACS Medicinal Chemistry Letters
Potent Neuronal Nicotinamide Adenine Dinucleotide-Boosting Tetrahydroquinoxalines: Structure-Activity Relationships and Early Drug Metabolism and Pharmacokinetics Evaluation
Experiments in human cellsInterventions